Synthesis and glycosidase inhibitory activity of 1-amino-3,6-anhydro-1-deoxy-D-sorbitol derivatives

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A tinglucal tributyl[4,6-O-bis(t-butyl)silylidene-3-O-tris(isopropyl)silyl]tin 7 and a triflate derived from isolevoglucosenone (1R,4R,5R)-4-benzyloxy-6,8-dioxabicyclo[3.2.1]oct-2-en-2-yl trifluoromethanesulfonate 10 undergo the carbonylative Stille conden ...

Synthesis and glycosidase inhibitory activity of 1-amino-3,6-anhydro-1-deoxy-D-sorbitol derivatives

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Generating macrocyclic inhibitors of protein-protein interactions

NICEdrug.ch, a workflow for rational drug design and systems-level analysis of drug metabolism

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SIRT2-and NRF2-Targeting Thiazole-Containing Compound with Therapeutic Activity in Huntington's Disease Models

Transferring lead-free piezoelectric ceramics into application

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Discovery of a Highly Tumor-Selective Organometallic Ruthenium(II)-Arene Complex

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Enumeration of 166 Billion Organic Small Molecules in the Chemical Universe Database GDB-17

Small Molecule Based Approaches to Inhibit Macrophage Migration Inhibitory Factor (MIF) Activities and Elucidate its Role in Health and Disease

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C(1 -> 4)-linked disaccharides through carbonylative Stille cross-coupling