Synthesis and glycosidase inhibitory activity of new penta-substituted C8-glycomimetics

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A one-pot, three-component synthesis of polysubstituted furo[2,3-c] quinoline 1 was developed based on the new reactivity profile of alpha-(4-nitrophenyl)-alpha-isocyanoacetates. Simply mixing aldehydes 2, ortho-alkynylanilines 3, and alpha-(4-nitrophenyl) ...

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Optimized protocols for the synthesis of diazolyl alpha,alpha-difluoroacetates via deoxofluorination of the corresponding glyoxylates with Morph-DAST are described. The method allowed the preparation of the title fluoridated building blocks in 73-96 % yiel ...

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This work presents a kinetic analysis of the exogenous photo-induced disinfection of E. coli in natural waters. Herein, the inactivation of bacteria by light and photo-generated transient species, i.e., hydroxyl radical (HO center dot), excited triplet sta ...

Synthesis and glycosidase inhibitory activity of new penta-substituted C8-glycomimetics

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Corrigendum to “Characterization of the glutathione redox state in the Golgi apparatus” [Redox Biol. 81 (2025) 103560]

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The domain of definition of the Levy white noise

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The emergence of crack-like behavior of frictional rupture: Edge singularity and energy balance

A solution method for predictive simulations in a stochastic environment

Synthesis and chemical transformations of diazolyl alpha,alpha-difluoroacetates

Decoding Neural Metabolic Markers From the Carotid Sinus Nerve in a Type 2 Diabetes Model

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The yeast C/D box snoRNA U14 adopts a "weak" K-turn like conformation recognized by the Snu13 core protein in solution

Kinetic modeling of lag times during photo-induced inactivation of E. coli in sunlit surface waters: Unraveling the pathways of exogenous action