Indole Alkaloids Synthesis via a Selective Cyclization of Aminocyclopropanes

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We report herein the enantioselective total synthesis of three monoterpene indole alkaloids, namely, (+)-alstilobanine C, (+)-undulifoline, and (-)-alpneumine H. The key features of our synthesis include: a) introduction of chirality via enantioselective d ...

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Indole Alkaloids Synthesis via a Selective Cyclization of Aminocyclopropanes

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New Strategies for the Functionalization of Alkenes Exploiting Tethering Chemistry and Ring Strain

Development of remote C-H bond functionalization of redox-active alcohol derivatives and oxidative transformations under photoredox catalysis

Nitrous oxide as a diazo transfer reagent: the synthesis of triazolopyridines

Natural Product Synthesis Enabled by Domino Processes Incorporating a 1,2-Rearrangement Step

New Vinylation and Alkynylation Strategies with Hypervalent Iodine Reagents and Diazo Compounds

Enantioselective Total Synthesis of (+)-Alstilobanine C, (+)-Undulifoline, and (-)-Alpneumine H

Tuning the π‐Accepting Properties of Mesoionic Carbenes: A Combined Computational and Experimental Study

Methods for the generation of large combinatorial macrocycle libraries

Isolation and characterization of diazoolefins

Copper‐Catalyzed Aza‐Sonogashira Cross‐Coupling to Ynimines: Development and Application to the Synthesis of Heterocycles