Publication

Strategy To Tether Organometallic Ruthenium-Arene Anticancer Compounds to Recombinant Human Serum Albumin

Publications associées (26)

Sustainable Hydrogenation of Nitroarenes to Anilines with Highly Active in-situ Generated Copper Nanoparticles

Mounir Driss Mensi, Berend Smit, Kyriakos Stylianou, Christopher Patrick Ireland, Ngoc Tú Nguyên, Fatma Pelin Uran

Metal nanoparticles (NPs) are usually stabilized by a capping agent, a surfactant, or a support material, to maintain their integrity. However, these strategies can impact their intrinsic catalytic activity. Here, we demonstrate that the in-situ formation ...

Wiley-VCH Verlag2020

DUBS: A Framework for Developing Directory of Useful Benchmarking Sets for Virtual Screening

Guillaume André Jean Fraux

Benchmarking is a crucial step in evaluating virtual screening methods for drug discovery. One major issue that arises among benchmarking data sets is a lack of a standardized format for representing the protein and ligand structures used to benchmark the ...

2020

Dual-Band Circularly Polarized Transmitarray Antenna for Satellite Communications at (20 to 30) GHz

Juan Ramon Mosig, Hamed Hasani, Joana Rita Alves dos Santos Silva, Maria Garcia Vigueras, Santiago Capdevila Cascante

A novel dual-band polarization-independent transmitarray is introduced in this paper for communication systems in Ka-band. Thanks to its unit-cell topology, the transmitarray antenna demonstrates almost complete independent performance at two design freque ...

2019

The virtuous cycle of human genetics and mouse models in drug discovery

Johan Auwerx

Ongoing studies in many species seek to understand the origins, architecture and consequences of phenotypic variation under normal and dysfunctional conditions, with the aim of identifying targets for intervention that can prevent, stabilize or reverse dis ...

NATURE PUBLISHING GROUP2019

Extrapolating the Fragment-Based Approach to Inorganic Drug Discovery

Paul Joseph Dyson, Lucinda Kate Batchelor

The fragment-based approach is a well-established strategy for organic drug discovery. Recent studies have shown that this approach also has considerable potential in medicinal inorganic chemistry, and yet the approach has not been formally described. Here ...

ELSEVIER2019

Innovative methods to release fine sediments from seasonal reservoirs

Giovanni De Cesare, Anton Schleiss, Pedro Filipe De Almeida Manso, Azin Amini, Sabine Chamoun, Sebastián Guillén Ludeña

The papers present three innovative solutions for fine sediment manage- ments in seasonal reservoirs, which are at different stages of maturity. Operational reservoir stirring using jet-like inflows may facilitate sediment routing, at no addi- tional cost ...

CRC Press/Balkema2018