Synthesis of Thiochromans via [3+3] Annulation of Aminocyclopropanes with Thiophenols

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Synthesis of Thiochromans via [3+3] Annulation of Aminocyclopropanes with Thiophenols

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Methods for high-throughput synthesis and screening of peptide libraries

Augmenting large language models with chemistry tools

Solid-phase peptide synthesis in 384-well plates

Go to the Board: A Journey through the Life of Professor David A. Evans

Enantio- and diastereoselective construction of vicinal C(sp(3)) centres via nickel-catalysed hydroalkylation of alkenes

Streamlined Alkylation via Nickel-Hydride-Catalyzed Hydrocarbonation of Alkenes

Ring-Opening Reactions of Aminocyclopropanes and Aminocyclobutanes

Modular Synthesis of Benzocyclobutenes via Pd(II)-Catalyzed Oxidative [2+2] Annulation of Arylboronic Acids with Alkenes

Chiral Alkyl Amine Synthesis via Catalytic Enantioselective Hydroalkylation of Enecarbamates

Methods for the generation of large combinatorial macrocycle libraries

Aliphatic Carboxylic Acids as Coupling Partners in Carbon-Heteroatom Bond-Forming Reactions

Development of Photocatalysts towards the Visible-Light driven C-Terminal Bioconjugation of Peptides and Proteins

Chiral Cyclopentadienyl Ligands: Design, Syntheses, and Applications in Asymmetric Catalysis

Synthesis and Characterization of Coordination Cages Based on Clathrochelate Metalloligands

Molecular nanostructures based on polyfunctional clathrochelate complexes

Development of cyclic peptide inhibitors of coagulation factor XII and matrix metalloproteinase 2

Decarboxylative C(sp3 )−O Cross-Coupling

Direct amidation of esters with nitroarenes

New methods for developing (bi)cyclic peptides by phage display

Elucidating the Role of Site-Specific Nitration of alpha-Synuclein in the Pathogenesis of Parkinson's Disease via Protein Semisynthesis and Mutagenesis